Monday, May 9, 2016

SERM effects

Tamoxifen: Inhibits breast tissue estrogen receptors, stimulates endometrial, stimulates bone. Endometrial hyperplasia side effect. Lowers total and LDL cholesterol, no effect on HDL. Used for premenopausal women.

Raloxifene: Inhibits breast tissue, inhibits endometrial, stimulates bone. No endometrial hyperplasia side effect. (So Relax!) used for postmenopausal women.

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